Targeted Therapy / Oncology & Neurology

Lemtrada (alemtuzumab)

Sanofi Genzyme · Anti-CD52 Monoclonal Antibody

FDA Approved 2014 Intravenous (IV) infusion Specialty Medication
Lemtrada alemtuzumab 12mg/1.2mL concentrate for infusion, Sanofi Genzyme, specialty pharmacy

What is Lemtrada? Lemtrada (alemtuzumab) is an anti-CD52 monoclonal antibody by Sanofi Genzyme. In oncology, alemtuzumab is used for B-cell chronic lymphocytic leukemia (CLL). The Lemtrada brand is approved for relapsing forms of multiple sclerosis (MS). A separate formulation (Campath) was previously marketed for CLL.

About Lemtrada

Brand NameLemtrada
Generic / INNalemtuzumab
Drug ClassAnti-CD52 Monoclonal Antibody
ManufacturerSanofi Genzyme
AdministrationIntravenous (IV) infusion
FDA Approval2014
📦 Lemtrada: 12 mg/1.2 mL (10 mg/mL) single-dose vials. Available ONLY through the Lemtrada REMS Program.

FDA-Approved Uses for Lemtrada

Indications are based on FDA approval. Your healthcare provider determines appropriate use based on your specific diagnosis, stage, biomarker status, and overall clinical picture.

  • Relapsing forms of multiple sclerosis (MS) — Lemtrada brand (when other therapies are inadequate)
  • B-cell chronic lymphocytic leukemia (CLL) — Campath brand (discontinued but alemtuzumab used under access programs)
Biomarker Note: No biomarker testing required for MS indication. For CLL (Campath), CD52 expression is universally high in B-CLL. Testing for TP53/del(17p) informs CLL treatment selection.

How Does Lemtrada Work?

Alemtuzumab targets CD52, a glycoprotein expressed on the surface of mature lymphocytes (B and T cells), monocytes, and NK cells. By binding CD52, alemtuzumab triggers complement-dependent cytotoxicity (CDC) and antibody-dependent cellular cytotoxicity (ADCC), depleting circulating lymphocytes and resetting the immune system.

Dosage & Administration

MS (Lemtrada): Two treatment courses — Course 1: 12 mg/day IV for 5 consecutive days; Course 2 (12 months later): 12 mg/day IV for 3 consecutive days. CLL (Campath/access programs): weight-based escalating doses per protocol.

⚠️ Important

Dosing is individualized by the prescribing clinician. Never adjust your dose without consulting your healthcare provider. This information is educational only and does not replace the official prescribing information.

Warnings, Precautions & Side Effects

General Warning

BOXED WARNINGS (Lemtrada): Autoimmune conditions (ITP — potentially fatal, nephropathies, thyroid disorders). Infusion reactions — severe and life-threatening. Malignancies — increased risk including thyroid cancer, melanoma, lymphoproliferative disorders. Lemtrada is only available through a REMS program due to these risks.

⛔ Serious Warnings & Precautions
  • Autoimmune ITP — potentially fatal (boxed)
  • Nephropathies (boxed)
  • Infusion reactions — life-threatening (boxed)
  • Secondary malignancies (boxed)
  • Life-threatening infections

Common Side Effects

  • Infusion reactions (rash, fever, urticaria)
  • Autoimmune thyroid disorders
  • Autoimmune ITP
  • Infections
  • Lymphopenia
  • Headache

This is not a complete list. Always report new or worsening symptoms to your healthcare provider promptly.

Storage & Handling

Refrigerate at 2°C to 8°C (36°F to 46°F). Do not freeze. Protect from light.

BiologicHealthPlus provides temperature-monitored cold-chain specialty delivery for medications requiring refrigeration. Never use a medication if its storage conditions have been compromised.

Insurance Coverage, Prior Authorization & Patient Assistance

🛡️ Commercial Insurance

Lemtrada is covered by most major commercial insurance plans when medically necessary and prior authorized. Coverage tier and cost-sharing vary by plan.

✅ Prior Authorization

Prior authorization is required by virtually all insurance plans for Lemtrada. BiologicHealthPlus handles the complete prior authorization process at no cost to patients or providers.

🏥 Medicare Coverage

Medicare Part B covers this IV medication when administered in a clinical setting. Medicaid coverage varies by state.

🆓 Patient Assistance

Manufacturer patient assistance programs may be available for eligible uninsured or underinsured patients. Contact BiologicHealthPlus for a confidential eligibility review.

Prior Authorization Patient Assistance Insurance & Savings Medication Costs

Frequently Asked Questions — Lemtrada

Lemtrada (alemtuzumab) is an anti-CD52 antibody approved for relapsing MS when other therapies have been inadequate. It depletes lymphocytes and resets the immune system. An older formulation (Campath) was used for CLL.

Because of serious risks including potentially fatal autoimmune conditions (ITP, nephropathies), severe infusion reactions, and secondary malignancies, Lemtrada is available only through certified healthcare facilities enrolled in the Lemtrada REMS program.

Intensive monitoring is required for at least 48 months after the last infusion — including monthly blood counts, kidney function, and thyroid function tests — to detect autoimmune complications early.

Related Medications

Calquence (acalabrutinib)  ·  Imbruvica (ibrutinib)  ·  Ocrevus (ocrelizumab — MS)  ·  Rituxan (rituximab)

Related Conditions

Relapsing multiple sclerosis (MS)  ·  Chronic lymphocytic leukemia (CLL)  ·  B-cell malignancies

Comparisons

Calquence

Authoritative References

Medical Disclaimer: This page is for general educational purposes only and does not constitute medical advice, diagnosis, or treatment. Always consult your oncologist, hematologist, or licensed healthcare professional before making any treatment decisions. Last reviewed: August 2026 by the BiologicHealthPlus Clinical Team.